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COVID answers in Scientific Journals all over the world


177 Results       Page 1

 [1] 
Elsevier: Antiviral Research
  original article Date Title Authors   Max. 6 Authors
1 [GO] 2024―Apr―09 Development of a highly stable, active small interfering RNA with broad activity against SARS-CoV viruses Beatrice Tolksdorf, Julian Heinze, Daniela Niemeyer, Viola Röhrs, Johanna Berg, Christian Drosten, Jens Kurreck
2 [GO] 2024―Mar―28 New conjugates based on N4-hydroxycytidine with more potent antiviral efficacy in vitro than EIDD-2801 against SARS-CoV-2 and other human coronaviruses Andrei E. Siniavin, Vladimir A. Gushchin, Natal'ya S. Shastina, Elizaveta S. Darnotuk, Sergey I. Luyksaar, Leonid I. Russu, Anna M. Inshakova, Elena V. Shidlovskaya, Daria V. Vasina, Nadezhda A. Kuznetsova, Daria M. Savina, Ilya D. Zorkov, Inna V. Dolzhikova, Anna B. Sheremet, Denis Y. Logunov, Nailya A. Zigangirova, Alexander L. Gintsburg
3 [GO] 2024―Mar―28 Azapeptides with unique covalent warheads as SARS-CoV-2 main protease inhibitors Kaustav Khatua, Yugendar R. Alugubelli, Kai S. Yang, Veerabhadra R. Vulupala, Lauren R. Blankenship, Demonta Coleman, Sandeep Atla, Sankar P. Chaki, Zhi Zachary Geng, Xinyu R. Ma, Jing Xiao, Peng-Hsun Chen, Chia-Chuan D. Cho, Shivangi Sharma, Erol C. Vatansever, Yuying Ma, Ge Yu, Benjamin W. Neuman, Shiqing Xu, Wenshe Ray Liu
4 [GO] 2024―Mar―14 A combination of nirmatrelvir and ombitasvir boosts inhibition of SARS-CoV-2 replication Christopher Moon, Eleanor Porges, Adam Roberts, Joanna Bacon
5 [GO] 2024―Mar―13 Caffeic acid phenethyl ester: An effective antiviral agent against porcine reproductive and Respiratory Syndrome Virus Zhanding Cui, Jing Zhang, Jinlong Wang, Jinlong Liu, Pu Sun, Jiaoyang Li, Guoxiu Li, Ying Sun, Juanbin Ying, Kun Li, Zhixun Zhao, Hong Yuan, Xingwen Bai, Xueqing Ma, Pinghua Li, Yuanfang Fu, Huifang Bao, Dong Li, Qiang Zhang, Zaixin Liu, Yimei Cao, Zengjun Lu
6 [GO] 2024―Mar―05 Glycan-directed SARS-CoV-2 inhibition by leek extract and lectins with insights into the mode-of-action of Concanavalin A Maja Klevanski, Heeyoung Kim, Mike Heilemann, Thomas Kuner, Ralf Bartenschlager
7 [GO] 2024―Mar―05 SARS-CoV-2 virus-like particle variants alpha and delta mimic the native viruses in their differential inflammasome activating potential Magdalena Bandyszewska, Magdalena Ambrożek-Latecka, Grażyna Hoser, Małgorzata Grzanka, Franziska Hornung, Stefanie Deinhardt-Emmer, Tomasz Skirecki
8 [GO] 2024―Mar―02 The host-targeted antiviral drug Zapnometinib exhibits a high barrier to the development of SARS-CoV-2 resistance André Schreiber, Franziska Rodner, Nicole Oberberg, Darisuren Anhlan, Stefan Bletz, Alexander Mellmann, Oliver Planz, Stephan Ludwig
9 [GO] 2024―Feb―28 Prophylactic effect of ensitrelvir in mice infected with SARS-CoV-2 Haruaki Nobori, Keiko Baba, Takayuki Kuroda, Kaoru Baba, Kazumi Matsumoto, Shinpei Yoshida, Ryosuke Watari, Yuki Tachibana, Teruhisa Kato, Keita Fukao
10 [GO] 2024―Feb―24 Methyl rosmarinate is an allosteric inhibitor of SARS-cov-2 3 C L protease as a potential candidate against SARS-cov-2 infection Hongtao Li, Meng Sun, Fuzhi Lei, Jinfeng Liu, Xixiang Chen, Yaqi Li, Ying Wang, Jiani Lu, Danmei Yu, Yueqiu Gao, Jianrong Xu, Hongzhuan Chen, Man Li, Zhigang Yi, Xiao He, Lili Chen
11 [GO] 2024―Feb―20 The α-dystroglycan N-terminus is a broad-spectrum antiviral agent against SARS-CoV-2 and enveloped viruses Maria Giulia Bigotti, Katja Klein, Esther S. Gan, Maria Anastasina, Simon Andersson, Olli Vapalahti, Pekka Katajisto, Maximilian Erdmann, Andrew D. Davidson, Sarah J. Butcher, Ian Collinson, Eng Eong Ooi, Giuseppe Balistreri, Andrea Brancaccio, Yohei Yamauchi
12 [GO] 2024―Feb―02 An adenovirus-vectored vaccine based on the N protein of feline coronavirus elicit robust protective immune responses Yuanhong Wang, Yun Liu, Junna Wang, Miao Zhang, Xiaoying Deng, Junhan Song, Jie Zhu, Lingxue Yu, Guoxin Li, Guangqing Liu
13 [GO] 2024―Feb―01 Therapeutic antibodies and alternative formats against SARS-CoV-2 Rahel R. Winiger, Laurent Perez
14 [GO] 2024―Jan―24 Drug repurposing platform for deciphering the druggable SARS-CoV-2 interactome Mariia S. Bogacheva, Suvi Kuivanen, Swapnil Potdar, Antti Hassinen, Sini Huuskonen, Ina Pöhner, Tamara J. Luck, Laura Turunen, Michaela Feodoroff, Leonora Szirovicza, Kirsi Savijoki, Jani Saarela, Päivi Tammela, Lassi Paavolainen, Antti Poso, Markku Varjosalo, Olli Kallioniemi, Vilja Pietiäinen, Olli Vapalahti
15 [GO] 2024―Jan―24 Generation and evaluation of protease inhibitor-resistant SARS-CoV-2 strains Hawa Sophia Bouzidi, Jean-Sélim Driouich, Raphaëlle Klitting, Ornéllie Bernadin, Géraldine Piorkowski, Rayane Amaral, Laurent Fraisse, Charles E. Mowbray, Ivan Scandale, Fanny Escudié, Eric Chatelain, Xavier de Lamballerie, Antoine Nougairède, Franck Touret
16 [GO] 2024―Jan―19 An intranasally delivered ultra-conserved siRNA prophylactically represses SARS-CoV-2 infection in the lung and nasal cavity. Adi Idris, Aroon Supramaniam, Yaman Tayyar, Gabrielle Kelly, NigelA.J. McMillan, Kevin V. Morris
17 [GO] 2024―Jan―09 TXM peptides inhibit SARS-CoV-2 infection, syncytia formation, and lower inflammatory consequences Tea Govednik, Duško Lainšček, Urška Kuhar, Marva Lachish, Sandra Janežič, Malan Štrbenc, Uroš Krapež, Roman Jerala, Daphne Atlas, Mateja Manček-Keber
18 [GO] 2023―Dec―27 A flexible, image-based, high-throughput platform encompassing in-depth cell profiling to identify broad-spectrum coronavirus antivirals with limited off-target effects Jordi Doijen, Inha Heo, Koen Temmerman, Peter Vermeulen, Annick Diels, Steffen Jaensch, Mark Burcin, Nick Van den Broeck, Valerie Raeymaekers, Joren Peremans, Katrien Konings, Maxime Clement, Danielle Peeters, Marnix Van Loock, Anil Koul, Christophe Buyck, Michiel Van Gool, Ellen Van Damme
19 [GO] 2023―Dec―27 Deubiquitinase USP39 promotes SARS-CoV-2 replication by deubiquitinating and stabilizing the envelope protein Xiang Chen, Li Tian, Linran Zhang, Wenying Gao, Miao Yu, Zhaolong Li, Wenyan Zhang
20 [GO] 2023―Dec―07 Nanobodies to multiple spike variants and inhalation of nanobody-containing aerosols neutralize SARS-CoV-2 in cell culture and hamsters Metin Aksu, Priya Kumar, Thomas Güttler, Waltraud Taxer, Kathrin Gregor, Bianka Mußil, Oleh Rymarenko, Kim M. Stegmann, Antje Dickmanns, Sabrina Gerber, Wencke Reineking, Claudia Schulz, Timo Henneck, Ahmed Mohamed, Gerhard Pohlmann, Mehmet Ramazanoglu, Kemal Mese, Uwe Groß, Tamar Ben-Yedidia, Oded Ovadia, Dalit Weinstein Fischer, Merav Kamensky, Amir Reichman, Wolfgang Baumgärtner, Maren von Köckritz-Blickwede, Matthias Dobbelstein, Dirk Görlich
21 [GO] 2023―Dec―05 Efficacy and safety of antiviral treatments for symptomatic COVID-19 outpatients: Systematic review and network meta-analysis Meital Zur, Thalia Peselev, Stav Yanko, Victoria Rotshild, Ilan Matok
22 [GO] 2023―Nov―30 Broad-spectrum antiviral activity of two structurally analogous CYP3A inhibitors against pathogenic human coronaviruses in vitro Lara Gallucci, James Bazire, Andrew D. Davidson, Iart Luca Shytaj
23 [GO] 2023―Nov―28 Oral delivery of a chitosan adjuvanted COVID-19 vaccine provides long-lasting and broad-spectrum protection against SARS-CoV-2 variants of concern in golden hamsters Shen Wang, Huan Cui, Cheng Zhang, Wujian Li, Weiqi Wang, Wenwen He, Na Feng, Yongkun Zhao, Tiecheng Wang, Xiaoqing Tang, Feihu Yan, Xianzhu Xia
24 [GO] 2023―Nov―24 A phenothiazine urea derivative broadly inhibits coronavirus replication via viral protease inhibition Katrina Forrestall, Eric S. Pringle, Dane Sands, Brett A. Duguay, Brett Farewell, Tekeleselassie Woldemariam, Darryl Falzarano, Ian Pottie, Craig McCormick, Sultan Darvesh
25 [GO] 2023―Nov―21 Lung transcriptomics of K18-hACE2 mice highlights mechanisms and genes involved in the MVA-S vaccine-mediated immune response and protection against SARS-CoV-2 infection Alberto Gómez-Carballa, Guillermo Albericio, Julián Montoto-Louzao, Patricia Pérez, David Astorgano, Irene Rivero-Calle, Federico Martinón-Torres, Mariano Esteban, Antonio Salas, Juan García-Arriaza
26 [GO] 2023―Nov―19 Monoglycosylated SARS-CoV-2 receptor binding domain fused with HAstem-scaffolded protein vaccine confers broad protective immunity against SARS-CoV-2 and influenza viruses Chia-Ying Wu, Yung-Chieh Tseng, Shao-En Kao, Li-Yang Wu, Jen-Tzu Hou, Yu-Chih Yang, Pei-Wen Hsiao, Juine-Ruey Chen
27 [GO] 2023―Nov―19 Newcastle Disease Virus (NDV)-based vaccine candidate against SARS-CoV-2 Omicron by intranasal immunization Qiu-Yan Zhang, Hong-Qing Zhang, Ya-Nan Zhang, Zhe-Rui Zhang, Xiao-Dan Li, Meng-Chan Hao, Yang Zhang, Jia-Qi Li, Yan-Yan Hu, Xiao-Ling Chen, Jing Wang, Yu-Jia Shi, Cheng-Lin Deng, Jian-Jun Chen, Han-Qing Ye, Bo Zhang
28 [GO] 2023―Nov―08 Fangchinoline inhibits SARS-CoV-2 and MERS-CoV entry Srikanth Sadhu, Jyotsna Dandotiya, Rajdeep Dalal, Ritika Khatri, Anna Z. Mykytyn, Aashima Batra, Manpreet Kaur, Rucha Chandwaskar, Virendra Singh, Aarzoo Kamboj, Mitul Srivastava, Shailendra Mani, Shailendra Asthana, Sweety Samal, Zaigham Abbas Rizvi, Deepak B. Salunke, Bart L. Haagmans, Amit Awasthi
29 [GO] 2023―Nov―08 Induction of neutralizing antibodies and mucosal IgA through intranasal immunization with the receptor binding domain of SARS-CoV-2 spike protein fused with the type IIb E. coli heat-labile enterotoxin A subunit He-Chin Hsieh, Chung-Chu Chen, Pin-Han Chou, Wen-Chun Liu, Suh-Chin Wu
30 [GO] 2023―Nov―08 A bivalent form of a RBD-specific synthetic antibody effectively neutralizes SARS-CoV-2 variants Dong-Gun Kim, Uijin Kim, In Ho Park, Bumhan Ryu, Youngki Yoo, Jeong Seok Cha, Ga-Yeon Yoon, Sung-Hee Kim, Heeju Oh, Jun-Young Seo, Ki Taek Nam, Je Kyung Seong, Jeon-Soo Shin, Hyun-Soo Cho, Hak-Sung Kim
31 [GO] 2023―Nov―07 Functional assessments of SARS-CoV-2 single-round infectious particles with variant-specific spike proteins on infectivity, drug sensitivity, and antibody neutralization Wen-Chi Su, Zan-Yu Chen, Young-Sheng Chang, King-Song Jeng, Uyen Nguyen Phuong Le, Yu-Chi Chou, Li-Lan Kuo, Ivonne Melano, Wei-Jan Wang, Ying-Chyi Song, Sin-Rong Li, Mien-Chie Hung, Michael M.C. Lai, Cheng-Wen Lin
32 [GO] 2023―Oct―18 Synthesis, evaluation, and mechanism of 1-(4-(arylethylenylcarbonyl)phenyl)-4-carboxy-2-pyrrolidinones as potent reversible SARS-CoV-2 entry inhibitors Srinivasa Rao Palla, Chen-Wei Li, Tai-Ling Chao, Hoi-Ling Vienn Lo, Liu Jia-Jin, Max Yu-Chen Pan, Yu-Ting Chiu, Wen-Chin Lin, Chih-Wei Hu, Chuen-Mi Yang, Yi-Ying Chen, Jun-Tung Fang, Sheng-Wei Lin, Yi-Tzu Lin, Hsiao-Ching Lin, Chih-Jung Kuo, Lily Hui-Ching Wang, Sui-Yuan Chang, Po-Huang Liang
33 [GO] 2023―Oct―18 ASK1 inhibitors are potential pan-antiviral drugs, which dampen replication of diverse viruses including SARS-CoV2 Wael L. Demian, Rajesh Abraham Jacob, Olga Cormier, Aisha Nazli, Matthew Melki, Akarin Asavajaru, Kaushal Baid, Ali Zhang, Matthew S. Miller, Charu Kaushic, Arinjay Banerjee, Karen Mossman
34 [GO] 2023―Oct―06 Induction of antiviral gene expression by cyclosporine a, but not inhibition of cyclophilin a or B, contributes to its restriction of human coronavirus 229E infection in a lung epithelial cell line John E. Mamatis, Carla E. Gallardo-Flores, Ujjwal Sangwan, Trinity H. Tooley, Taylor Walsh, Che C. Colpitts
35 [GO] 2023―Sep―28 Corrigendum to ’ Sangivamycin is preferentially incorporated into viral RNA by the SARS-CoV-2 polymerase’ [Antiviral Research 218 (2023) 105716-105728/ doi: 10.1016/j.antiviral.2023.105716] Ryan P. Bennett, Yasemin Yoluç, Jason D. Salter, Alexander Ripp, Henning J. Jessen, Stefanie M. Kaiser, Harold C. Smith
36 [GO] 2023―Sep―09 Sangivamycin is preferentially incorporated into viral RNA by the SARS-CoV-2 polymerase Ryan P. Bennett, Yasemin Yoluç, Jason D. Salter, Alexander Ripp, Henning J. Jessen, Stefanie M. Kaiser, Harold C. Smith
37 [GO] 2023―Aug―09 Diketo acid inhibitors of nsp13 of SARS-CoV-2 block viral replication Angela Corona, Valentina Noemi Madia, Riccardo De Santis, Candida Manelfi, Roberta Emmolo, Davide Ialongo, Elisa Patacchini, Antonella Messore, Donatella Amatore, Giovanni Faggioni, Marco Artico, Daniela Iaconis, Carmine Talarico, Roberto Di Santo, Florigio Lista, Roberta Costi, Enzo Tramontano
38 [GO] 2023―Aug―09 PRO-2000 exhibits SARS-CoV-2 antiviral activity by interfering with spike-heparin binding Evelien Vanderlinden, Arnaud Boonen, Sam Noppen, Geert Schoofs, Maya Imbrechts, Nick Geukens, Robert Snoeck, Annelies Stevaert, Lieve Naesens, Graciela Andrei, Dominique Schols
39 [GO] 2023―Jul―20 Novel siRNA therapeutics demonstrate multi-variant efficacy against SARS-CoV-2 Ellen Bowden-Reid, Scott Ledger, Yuan Zhang, Francesca Di Giallonardo, Anupriya Aggarwal, Alberto Ospina Stella, Anouschka Akerman, Vanessa Milogiannakis, Gregory Walker, William Rawlinson, Stuart Turville, Anthony D. Kelleher, Chantelle Ahlenstiel
40 [GO] 2023―Jul―20 Ceragenins exhibit antiviral activity against SARS-CoV-2 by increasing the expression and release of type I interferons upon activation of the host's immune response Łukasz Suprewicz, Artur Szczepański, Marzena Lenart, Ewelina Piktel, Krzysztof Fiedoruk, Emilia Barreto-Duran, Anna Kula-Pacurar, Paul B. Savage, Aleksandra Milewska, Robert Bucki, Krzysztof Pyrć
41 [GO] 2023―Jul―17 Seasonal coronavirus infections trigger NLRP3 inflammasome activation in macrophages but is therapeutically targetable Yang Li, Yining Wang, Yunlong Li, Annemarie C. de Vries, Pengfei Li, Maikel P. Peppelenbosch, Qiuwei Pan
42 [GO] 2023―Jul―13 Assessment of the frequency of SARS-CoV-2 Omicron variant escape from RNA-dependent RNA polymerase inhibitors and 3C-like protease inhibitors Emi Takashita, Seiichiro Fujisaki, Hiroko Morita, Shiho Nagata, Hideka Miura, Mami Nagashima, Shinji Watanabe, Makoto Takeda, Yoshihiro Kawaoka, Hideki Hasegawa
43 [GO] 2023―Jul―11 Evaluating Z-FA-FMK, a host cathepsin L protease inhibitor, as a potent and broad-spectrum antiviral therapy against SARS-CoV-2 and related coronaviruses Ju Hwan Jeong, Jang-Hoon Choi, Beom Kyu Kim, Seong Cheol Min, Santosh Chokkakula, Sol Oh, Ji-Hyun Park, Sang-Mu Shim, Eung-Gook Kim, Young Ki Choi, Joo-Yeon Lee, Yun Hee Baek, Min-Suk Song
44 [GO] 2023―Jul―08 Identification of alpha-linolenic acid as a broad-spectrum antiviral against zika, dengue, herpes simplex, influenza virus and SARS-CoV-2 infection Yifei Feng, Yan Yang, Shuting Zou, Shuqi Qiu, Hao Yang, Yi Hu, Guifen Lin, Xingang Yao, Shuwen Liu, Min Zou
45 [GO] 2023―Jun―25 Paxlovid for hospitalized COVID-19 patients with chronic kidney disease Hong Cai, Jiayi Yan, Shang Liu, Ping Li, Li Ding, Yaping Zhan, Jiayue Lu, Zhenyuan Li, Mingli Zhu, Yuan Gao, XingRong Gong, Haiqun Ban, Leyi Gu, Weibin Zhou, Jieying Wang, Shan Mou
46 [GO] 2023―Jun―23 Cathepsin inhibitors nitroxoline and its derivatives inhibit SARS-CoV-2 infection Rafaela Milan Bonotto, Ana Mitrović, Izidor Sosič, Pamela Martinez-Orellana, Federica Dattola, Stanislav Gobec, Janko Kos, Alessandro Marcello
47 [GO] 2023―Jun―15 Intranasal delivery of an adenovirus-vector vaccine co-expressing a modified spike protein and a genetic adjuvant confers lasting mucosal immunity against SARS-CoV-2 Hi Eun Jung, Keun Bon Ku, Byeong Hoon Kang, Jang Hyun Park, Hyeon Cheol Kim, Kyun-Do Kim, Heung Kyu Lee
48 [GO] 2023―Jun―15 Combining virtual screening with cis-/trans-cleavage enzymatic assays effectively reveals broad-spectrum inhibitors that target the main proteases of SARS-CoV-2 and MERS-CoV Yu-Jen Chang, Uyen Nguyen Phuong Le, Jia-Jun Liu, Sin-Rong Li, Shao-Ting Chao, Hsueh-Chou Lai, Yu-Feng Lin, Kai-Cheng Hsu, Chih-Hao Lu, Cheng-Wen Lin
49 [GO] 2023―May―18 SARS-CoV-2 induces cardiomyocyte apoptosis and inflammation but can be ameliorated by ACE inhibitor Captopril Xiaohan Huang, Wenxia Fan, Jing Sun, Jiaqing Yang, Yanjun Zhang, Qian Wang, Pingchao Li, Yudi Zhang, Shengnan Zhang, Heying Li, Jianhua Wang, Liqiang Feng, Jincun Zhao, Ling Chen, Qu Linbing
50 [GO] 2023―Apr―20 Evaluation of antiviral drugs against newly emerged SARS-CoV-2 Omicron subvariants Junhyung Cho, Younmin Shin, Jeong-Sun Yang, Jun Won Kim, Kyung-Chang Kim, Joo-Yeon Lee
51 [GO] 2023―Apr―18 Omicsynin B4 potently blocks coronavirus infection by inhibiting host proteases cathepsin L and TMPRSS2 Yihua Li, Kun Wang, Hongmin Sun, Shuo Wu, Huiqiang Wang, Yuanyuan Shi, Xingxing Li, Haiyan Yan, Ge Yang, Mengyuan Wu, Yihong Li, Xiaotian Ding, Shuyi Si, Jiandong Jiang, Yu Du, Yuhuan Li, Bin Hong
52 [GO] 2023―Apr―15 Longitudinal analyses using 18F-Fluorodeoxyglucose positron emission tomography with computed tomography as a measure of COVID-19 severity in the aged, young, and humanized ACE2 SARS-CoV-2 hamster models Yu Cong, Ji Hyun Lee, Donna L. Perry, Kurt Cooper, Hui Wang, Saurabh Dixit, David X. Liu, Irwin M. Feuerstein, Jeffrey Solomon, Christopher Bartos, Jurgen Seidel, Dima A. Hammoud, Ricky Adams, Scott M. Anthony, Janie Liang, Nicolette Schuko, Rong Li, Yanan Liu, Zhongde Wang, E. Bart Tarbet, Amanda M.W. Hischak, Randy Hart, Nejra Isic, Tracey Burdette, David Drawbaugh, Louis M. Huzella, Russell Byrum, Danny Ragland, Marisa C. St Claire, Jiro Wada, Jonathan R. Kurtz, Lisa E. Hensley, Connie S. Schmaljohn, Michael R. Holbrook, Reed F. Johnson
53 [GO] 2023―Mar―31 The multiple roles of nsp6 in the molecular pathogenesis of SARS-CoV-2 Cody Bills, Xuping Xie, Pei-Yong Shi
54 [GO] 2023―Mar―30 Evaluation of a panel of therapeutic antibody clinical candidates for efficacy against SARS-CoV-2 in Syrian hamsters Yu Cong, Eric M. Mucker, Donna L. Perry, Saurabh Dixit, Erin Kollins, Russ Byrum, Louis Huzella, Robert Kim, Mathew Josleyn, Steven Kwilas, Christopher Stefan, Charles J. Shoemaker, Jeff Koehler, Susan Coyne, Korey Delp, Janie Liang, David Drawbaugh, Amanda Hischak, Randy Hart, Elena Postnikova, Nick Vaughan, Jason Asher, Marisa St Claire, Jarod Hanson, Connie Schmaljohn, Ann E. Eakin, Jay W. Hooper, Michael R. Holbrook
55 [GO] 2023―Mar―28 Synthesis of deuterated S-217622 (Ensitrelvir) with antiviral activity against coronaviruses including SARS-CoV-2 Yujian Yang, Liu Cao, Ming Yan, Jun Zhou, Sidi Yang, Tiefeng Xu, Siyao Huang, Kun Li, Qifan Zhou, Guanguan Li, Yujun Zhu, Feng Cong, Hongmin Zhang, Deyin Guo, Yingjun Li, Xumu Zhang
56 [GO] 2023―Mar―26 Cellular electrical impedance to profile SARS-CoV-2 fusion inhibitors and to assess the fusogenic potential of spike mutants Emiel Vanhulle, Jordi Doijen, Joren Stroobants, Becky Provinciael, Sam Noppen, Dominique Schols, Annelies Stevaert, Kurt Vermeire
57 [GO] 2023―Mar―20 SARS-CoV-2 Omicron (B.1.1.529) shows minimal neurotropism in a double-humanized mouse model Rubens Prince dos Santos Alves, Ying-Ting Wang, Zbigniew Mikulski, Sara McArdle, Norazizah Shafee, Kristen M. Valentine, Robyn Miller, Shailendra Verma, Fernanda Ana Sosa Batiz, Erin Maule, Michael N. Nguyen, Julia Timis, Colin Mann, Michelle Zandonatti, Suzie Alarcon, Jenny Rowe, Mitchell Kronenberg, Daniela Weiskopf, Alessandro Sette, Kathryn Hastie, Erica Ollmann Saphire, Stephen Festin, Kenneth Kim, Sujan Shresta
58 [GO] 2023―Mar―05 Heterologous boost with mRNA vaccines against SARS-CoV-2 Delta/Omicron variants following an inactivated whole-virus vaccine Changrui Lu, Yuntao Zhang, Xiaohu Liu, Fujun Hou, Rujie Cai, Zhibin Yu, Fei Liu, Guohuan Yang, Jun Ding, Jiang Xu, Xianwu Hua, Xinhua Cheng, Xinping Pan, Lianxiao Liu, Kang Lin, Zejun Wang, Xinguo Li, Jia Lu, Qiu Zhang, Yuwei Li, Chunxia Hu, Huifen Fan, Xiaoke Liu, Hui Wang, Rui Jia, Fangjingwei Xu, Xuewei Wang, Hongwei Huang, Ronghua Zhao, Jing Li, Hang Cheng, William Jia, Xiaoming Yang
59 [GO] 2023―Mar―02 Cyclic lipopeptides as membrane fusion inhibitors against SARS-CoV-2: New tricks for old dogs Egor V. Shekunov, Polina D. Zlodeeva, Svetlana S. Efimova, Anna A. Muryleva, Vladimir V. Zarubaev, Alexander V. Slita, Olga S. Ostroumova
60 [GO] 2023―Mar―02 Novel bispecific human antibody platform specifically targeting a fully open spike conformation potently neutralizes multiple SARS-CoV-2 variants Ji Woong Kim, Kyun Heo, Hyun Jung Kim, Youngki Yoo, Hyun-Soo Cho, Hui Jeong Jang, Ho-Young Lee, In Young Ko, Ju Rang Woo, Yea Bin Cho, Ji Hyun Lee, Ha Rim Yang, Ha Gyeong Shin, Hye Lim Choi, Kyusang Hwang, Sokho Kim, Hanseong Kim, Kwangrok Chun, Sukmook Lee
61 [GO] 2023―Mar―01 Pinosrtobin from plants and propolis against human coronavirus HCoV-OC43 by modulating host AHR/CYP1A1 pathway and lipid metabolism Liyun Zhao, Liyuan Yao, Rui Chen, Jiani He, Tingting Lin, Silin Qiu, Guohua Chen, Hongfeng Chen, Sheng-Xiang Qiu
62 [GO] 2023―Mar―01 Design and characterization of novel SARS-CoV-2 fusion inhibitors with N-terminally extended HR2 peptides Yue Hu, Yuanmei Zhu, Yanying Yu, Nian Liu, Xiaohui Ju, Qiang Ding, Yuxian He
63 [GO] 2023―Feb―18 CDK4/6 inhibitor palbociclib promotes SARS-CoV-2 cell entry by down-regulating SKP2 dependent ACE2 degradation Yingzi Xiao, Ying Yan, Le Chang, Huimin Ji, Huizhen Sun, Shi Song, Kaihao Feng, Abudulimutailipu Nuermaimaiti, Zhuoqun Lu, Lunan Wang
64 [GO] 2023―Feb―14 Nirmatrelvir exerts distinct antiviral potency against different human coronaviruses Jiajing Li, Yining Wang, Kundan Solanki, Rajat Atre, Marla Lavrijsen, Qiuwei Pan, Mirza S. Baig, Pengfei Li
65 [GO] 2023―Feb―03 Nucleolin mediates SARS-CoV-2 replication and viral-induced apoptosis of host cells Vanessa F. Merino, Yu Yan, Alvaro A. Ordonez, C. Korin Bullen, Albert Lee, Harumi Saeki, Krishanu Ray, Tao Huang, Sanjay K. Jain, Martin G. Pomper
66 [GO] 2023―Jan―20 Development of highly effective LCB1-based lipopeptides targeting the spike receptor-binding motif of SARS-CoV-2 Yuanmei Zhu, Min Li, Nian Liu, Tong Wu, Xuelian Han, Guangyu Zhao, Yuxian He
67 [GO] 2022―Dec―29 “Flavivirus proteases: The viral Achilles heel to prevent future pandemics” Tadahisa Teramoto, Kyung H. Choi, Radhakrishnan Padmanabhan
68 [GO] 2022―Dec―27 Targeting SARS-CoV-2 and host cell receptor interactions Siew Pheng Lim
69 [GO] 2022―Dec―24 A new intracellular targeting motif in the cytoplasmic tail of the spike protein may act as a target to inhibit SARS-CoV-2 assembly Longbo Hu, Yongjie Tang, Lingling Mei, Mengdi Liang, Jinxian Huang, Xufei Wang, Liping Wu, Jiajing Jiang, Leyi Li, Fei Long, Jing Xiao, Long Tan, Shaohua Lu, Tao Peng
70 [GO] 2022―Dec―23 Influenza antivirals and their role in pandemic preparedness Jeremy C. Jones, Hui-Ling Yen, Peter Adams, Kimberly Armstrong, Elena A. Govorkova
71 [GO] 2022―Dec―22 Kill or corrupt: Mechanisms of action and drug-resistance of nucleotide analogues against SARS-CoV-2 Ashleigh Shannon, Bruno Canard
72 [GO] 2022―Dec―22 Reverse genetic systems of SARS-CoV-2 for antiviral research Chaitanya Kurhade, Xuping Xie, Pei-Yong Shi
73 [GO] 2022―Dec―21 Intranasal delivery of replicating mRNA encoding hACE2-targeting antibody against SARS-CoV-2 Omicron infection in the hamster Ya-Nan Zhang, Hong-Qing Zhang, Gui-Feng Wang, Zhe-Rui Zhang, Jia-Qi Li, Xiao-Ling Chen, Yan-Yan Hu, Xiang-Yue Zeng, Yu-Jia Shi, Jing Wang, Ying-Hua Li, Xiao-Dan Li, Chun-He Wang, Bing Zhu, Bo Zhang
74 [GO] 2022―Dec―21 Development of a robust and convenient dual-reporter high-throughput screening assay for SARS-CoV-2 antiviral drug discovery Winston Chiu, Joost Schepers, Thibault Francken, Laura Vangeel, Kayvan Abbasi, Dirk Jochmans, Steven De Jonghe, Hendrik Jan Thibaut, Volker Thiel, Johan Neyts, Manon Laporte, Pieter Leyssen
75 [GO] 2022―Dec―16 Evaluation of molnupiravir (EIDD-2801) efficacy against SARS-CoV-2 in the rhesus macaque model Dylan M. Johnson, Trevor Brasel, Shane Massey, Tania Garron, Michael Grimes, Jeanon Smith, Maricela Torres, Shannon Wallace, Alejandro Villasante-Tezanos, David W. Beasley, Jason E. Comer
76 [GO] 2022―Dec―05 Phenothiazines inhibit SARS-CoV-2 cell entry via a blockade of spike protein binding to neuropilin-1 Mei Hashizume, Ayako Takashima, Chikako Ono, Toru Okamoto, Masaharu Iwasaki
77 [GO] 2022―Dec―01 RBM24 inhibits the translation of SARS-CoV-2 polyproteins by targeting the 5ʹ-untranslated region Yongxuan Yao, Hao Sun, Yingshan Chen, Lingqian Tian, Dan Huang, Canyu Liu, Yuan Zhou, Yun Wang, Zhe Wen, Bo Yang, Xinwen Chen, Rongjuan Pei
78 [GO] 2022―Nov―23 Rapid discovery and classification of inhibitors of coronavirus infection by pseudovirus screen and amplified luminescence proximity homogeneous assay Kwiwan Jeong, JuOae Chang, Sun-mi Park, Jinhee Kim, Sangeun Jeon, Dong Hwan Kim, Young-Eui Kim, Joo Chan Lee, Somyoung Im, Yejin Jo, Ji-Young Min, Hanbyeul Lee, Minjoo Yeom, Sang-Hyuk Seok, Da In On, Hyuna Noh, Jun-Won Yun, Jun Won Park, Daesub Song, Je Kyung Seong, Kyung-Chang Kim, Joo-Yeon Lee, Hyun-Ju Park, Seungtaek Kim, Tae-gyu Nam, Wonsik Lee
79 [GO] 2022―Nov―21 Inhibition of p38 signaling curtails the SARS-CoV-2 induced inflammatory response but retains the IFN-dependent antiviral defense of the lung epithelial barrier Aileen Faist, Sebastian Schloer, Angeles Mecate-Zambrano, Josua Janowski, André Schreiber, Yvonne Boergeling, Beate C.G. Conrad, Sriram Kumar, Leonie Toebben, Klaus Schughart, Morris Baumgardt, Mirjana Kessler, Katja Hoenzke, Andreas Hocke, Marcel Trautmann, Wolfgang Hartmann, Hiroki Kato, Ursula Rescher, Anmari Christersson, Joachim Kuehn, Alexander Mellmann, Thorsten Wolff, Philip Kuempers, Alexandros Rovas, Rainer Wiewrodt, Karsten Wiebe, Peter Barth, Stephan Ludwig, Linda Brunotte
80 [GO] 2022―Nov―17 In vitro and in vivo effects of 3-indoleacetonitrile-A potential new broad-spectrum therapeutic agent for SARS-CoV-2 infection Xianfeng Hui, Xiao Yu, Kun Huang, Ting Xu, Lei Cao, Yufei Zhang, Lianzhong Zhao, Ya Zhao, Changjie Lv, sheng Feng, Yongzhong Jiang, Linlin Liu, Meilin Jin
81 [GO] 2022―Nov―03 Structure and inhibition of SARS-CoV-1 and SARS-CoV-2 main proteases by oral antiviral compound AG7404 Montserrat Fàbrega-Ferrer, Alejandra Herrera-Morandé, Sara Muriel-Goñi, Julia Pérez-Saavedra, Paula Bueno, Victoria Castro, Urtzi Garaigorta, Pablo Gastaminza, Miquel Coll
82 [GO] 2022―Oct―31 Topoisomerase 3b is dispensable for replication of a positive-sense RNA virus--murine coronavirus Tianyi Zhang, Shuaikun Su, Valerie Altouma, Xingliang Zhu, Yutong Xue, Weiping Shen, Brian Wilgenburg, Weidong Wang
83 [GO] 2022―Oct―30 In vitro and in vivo evaluation of the main protease inhibitor FB2001 against SARS-CoV-2 Weijuan Shang, Wenhao Dai, Cheng Yao, Ling Xu, Xiangming Tao, Haixia Su, Jian Li, Xiong Xie, Yechun Xu, Min Hu, Dong Xie, Hualiang Jiang, Leike Zhang, Hong Liu
84 [GO] 2022―Oct―29 Geneticin shows selective antiviral activity against SARS-CoV-2 by interfering with programmed -1 ribosomal frameshifting Carmine Varricchio, Gregory Mathez, Trestan Pillonel, Claire Bertelli, Laurent Kaiser, Caroline Tapparel, Andrea Brancale, Valeria Cagno
85 [GO] 2022―Oct―17 Potent inhibition of diverse Omicron sublineages by SARS-CoV-2 fusion-inhibitory lipopeptides Yuanmei Zhu, Yue Hu, Nian Liu, Huihui Chong, Yuxian He
86 [GO] 2022―Oct―15 Astersaponin I from Aster koraiensis is a natural viral fusion blocker that inhibit the infection of SARS-CoV-2 variants and syncytium formation Tai Young Kim, Ji-Young Kim, Hak Cheol Kwon, Sangeun Jeon, Sol ji Lee, Haejin Jung, Seungtaek Kim, Dae Sik Jang, C Justin Lee
87 [GO] 2022―Oct―06 Combination therapy with nirmatrelvir and molnupiravir improves the survival of SARS-CoV-2 infected mice Ju Hwan Jeong, Santosh Chokkakula, Seong Cheol Min, Beom Kyu Kim, Won-Suk Choi, Sol Oh, Yu Soo Yun, Da Hyeon Kang, Ok-Jun Lee, Eung-Gook Kim, Jang-Hoon Choi, Joo-Yeon Lee, Young Ki Choi, Yun Hee Baek, Min-Suk Song
88 [GO] 2022―Oct―05 Generation of a VeroE6 Pgp gene knock out cell line and its use in SARS-CoV-2 antiviral study Yuao Zhu, Joe Binder, Irina Yurgelonis, Devendra Rai, Sarah Lazarro, Chester Costales, Keith Kobylarz, Patricia McMonagle, Claire M. Steppan, Lisa Aschenbrenner, Annaliesa S. Anderson, Rhonda D. Cardin
89 [GO] 2022―Sep―23 Repurposing of HIV/HCV protease inhibitors against SARS-CoV-2 3CLpro Ling Ma, Quanjie Li, Yongli Xie, Dongrong Yi, Saisai Guo, Fei Guo, Jing Wang, Long Yang, Shan Cen
90 [GO] 2022―Aug―28 Brequinar and dipyridamole in combination exhibits synergistic antiviral activity against SARS-CoV-2 in vitro: Rationale for a host-acting antiviral treatment strategy for COVID-19 James F. Demarest, Maryline Kienle, RuthMabel Boytz, Mary Ayres, Eun Jung Kim, Justin J. Patten, Donghoon Chung, Varsha Gandhi, Robert Davey, David B. Sykes, Nadim Shohdy, John C. Pottage, Vikram S. Kumar
91 [GO] 2022―Aug―17 Punicalagin as an allosteric NSP13 helicase inhibitor potently suppresses SARS-CoV-2 replication in vitro Lian Lu, Yun Peng, Huiqiao Yao, Yanqun Wang, Jinyu Li, Yang Yang, Zhonghui Lin
92 [GO] 2022―Jul―31 Rational design of AAVrh10-vectored ACE2 functional domain to broadly block the cell entry of SARS-CoV-2 variants Minchao Li, Jiaoshan Chen, Yajie Liu, Jin Zhao, Yanjun Li, Yunqi Hu, Yaoqing Chen, Litao Sun, Yuelong Shu, Fengling Feng, Caijun Sun
93 [GO] 2022―Jul―11 Allosteric inhibitors of the main protease of SARS-CoV-2 Subodh Kumar Samrat, Jimin Xu, Xuping Xie, Eleonora Gianti, Haiying Chen, Jing Zou, Jason G. Pattis, Khaled Elokely, Hyun Lee, Zhong Li, Michael L. Klein, Pei-Yong Shi, Jia Zhou, Hongmin Li
94 [GO] 2022―Jul―04 Different efficacies of neutralizing antibodies and antiviral drugs on SARS-CoV-2 Omicron subvariants, BA.1 and BA.2 Hirofumi Ohashi, Takayuki Hishiki, Daisuke Akazawa, Kwang Su Kim, Joohyeon Woo, Kaho Shionoya, Kana Tsuchimoto, Shoya Iwanami, Saya Moriyama, Hitomi Kinoshita, Souichi Yamada, Yudai Kuroda, Tsukasa Yamamoto, Noriko Kishida, Shinji Watanabe, Hideki Hasegawa, Hideki Ebihara, Tadaki Suzuki, Maeda Ken, Shuetsu Fukushi, Yoshimasa Takahashi, Shingo Iwami, Koichi Watashi
95 [GO] 2022―Jul―04 Hydroxypropyl-beta-cyclodextrin (HP-BCD) inhibits SARS-CoV-2 replication and virus-induced inflammatory cytokines Bruno Braz Bezerra, Gustavo Peixoto Duarte da Silva, Sharton Vinicius Antunes Coelho, Isadora Alonso Correa, Marcos Romario Matos de Souza, Keylla Vitória Gomes Macedo, Bruna Machado Matos, Amilcar Tanuri, Flavio Lemos Matassoli, Luciana Jesus da Costa, James E.K. Hildreth, Luciana Barros de Arruda
96 [GO] 2022―Jun―29 Inhibition of a broad range of SARS-CoV-2 variants by antiviral phytochemicals in hACE2 mice Eun-Ha Kim, Ba Wool Lee, Byeol Ryu, Hyo Moon Cho, Se-Mi Kim, Seung-Gyu Jang, Mark Anthony B. Casel, Rare Rollon, Ji-Seung Yoo, Haryoung Poo, Won Keun Oh, Young Ki Choi
97 [GO] 2022―Jun―27 A circular mRNA vaccine prototype producing VFLIP-X spike confers a broad neutralization of SARS-CoV-2 variants by mouse sera Chotiwat Seephetdee, Kanit Bhukhai, Nattawut Buasri, Puttipatch Leelukkanaveera, Pat Lerdwattanasombat, Suwimon Manopwisedjaroen, Nut Phueakphud, Sakonwan Kuhaudomlarp, Eduardo Olmedillas, Erica Ollmann Saphire, Arunee Thitithanyanont, Suradej Hongeng, Patompon Wongtrakoongate
98 [GO] 2022―Jun―21 Numb-associated kinases are required for SARS-CoV-2 infection and are cellular targets for antiviral strategies Marwah Karim, Sirle Saul, Luca Ghita, Malaya Kumar Sahoo, Chengjin Ye, Nishank Bhalla, Chieh Wen Lo, Jing Jin, Jun-Gyu Park, Belén Martinez-Gualda, Michael Patrick East, Gary L. Johnson, Benjamin A. Pinsky, Luis Martinez-Sobrido, Christopher R.M. Asquith, Aarthi Narayanan, Steven De Jonghe, Shirit Einav
99 [GO] 2022―Jun―19 Bergamottin, a bioactive component of bergamot, inhibits SARS-CoV-2 infection in golden Syrian hamsters Minmin Zhou, Yang Liu, Junyuan Cao, Siqi Dong, Yuxia Hou, Yan Yu, Qiuyan Zhang, Yueli Zhang, Xiaoying Jia, Bo Zhang, Gengfu Xiao, Gang Li, Wei Wang
100 [GO] 2022―Jun―16 Identification of potent inhibitors of arenavirus and SARS-CoV-2 exoribonucleases by fluorescence polarization assay Sergio Hernández, Mikael Feracci, Carolina Trajano De Jesus, Priscila El Kazzi, Rafik Kaci, Laura Garlatti, Clemence Mondielli, Fabrice Bailly, Philippe Cotelle, Franck Touret, Xavier de Lamballerie, Bruno Coutard, Etienne Decroly, Bruno Canard, François Ferron, Karine Alvarez
101 [GO] 2022―Jun―10 Conserved coronavirus proteins as targets of broad-spectrum antivirals Cleber C. Melo-Filho, Tesia Bobrowski, Holli-Joi Martin, Zoe Sessions, Konstantin Popov, Nathaniel J. Moorman, Ralph S. Baric, Eugene N. Muratov, Alexander Tropsha
102 [GO] 2022―Jun―07 Discovery of novel SARS-CoV-2 inhibitors targeting the main protease Mpro by virtual screenings and hit optimization Beatrice Mercorelli, Jenny Desantis, Marta Celegato, Alessandro Bazzacco, Lydia Siragusa, Paolo Benedetti, Michela Eleuteri, Federico Croci, Gabriele Cruciani, Laura Goracci, Arianna Loregian
103 [GO] 2022―May―28 A novel high-throughput single B-cell cloning platform for isolation and characterization of high-affinity and potent SARS-CoV-2 neutralizing antibodies Paritosh Prashar, Sonali Swain, Nisha Adhikari, Punit Aryan, Anupama Singh, Mohit Kwatra, Prabhakar B
104 [GO] 2022―May―21 Animal models for studying coronavirus infections and developing antiviral agents and vaccines Qisheng Lin, Chunni Lu, Yuqi Hong, Runfeng Li, Jinding Chen, Weisan Chen, Jianxin Chen
105 [GO] 2022―May―19 Immunodetection assays for the quantification of seasonal common cold coronaviruses OC43, NL63, or 229E infection confirm nirmatrelvir as broad coronavirus inhibitor Tatjana Weil, Jan Lawrenz, Alina Seidel, Jan Münch, Janis A. Müller
106 [GO] 2022―May―19 Discovery of compounds that inhibit SARS-CoV-2 Mac1-ADP-ribose binding by high-throughput screening Anu Roy, Yousef M. Alhammad, Peter McDonald, David K. Johnson, Junlin Zhuo, Sarah Wazir, Dana Ferraris, Lari Lehtiö, Anthony K.L. Leung, Anthony R. Fehr
107 [GO] 2022―May―18 SARS-CoV-2 Permissive glioblastoma cell line for high throughput antiviral screening Emiel Vanhulle, Joren Stroobants, Becky Provinciael, Anita Camps, Sam Noppen, Piet Maes, Kurt Vermeire
108 [GO] 2022―May―07 Development of a cost-effective ovine antibody-based therapy against SARS-CoV-2 infection and contribution of antibodies specific to the spike subunit proteins Stephen Findlay-Wilson, Linda Easterbrook, Sandra Smith, Neville Pope, Gareth Humphries, Holger Schuhmann, Didier Ngabo, Emma Rayner, Ashley David Otter, Tom Coleman, Bethany Hicks, Victoria Anne Graham, Rachel Halkerston, Kostis Apostolakis, Stephen Taylor, Susan Fotheringham, Amanda Horton, Julia Anne Tree, Matthew Wand, Roger Hewson, Stuart David Dowall
109 [GO] 2022―May―05 Intravenous delivery of GS-441524 is efficacious in the African green monkey model of SARS-CoV-2 infection Jared Pitts, Darius Babusis, Meghan S. Vermillion, Raju Subramanian, Kim Barrett, Diane Lye, Bin Ma, Xiaofeng Zhao, Nicholas Riola, Xuping Xie, Adriana Kajon, Xianghan Lu, Roy Bannister, Pei-Yong Shi, Maria Toteva, Danielle P. Porter, Bill J. Smith, Tomas Cihlar, Richard Mackman, John P. Bilello
110 [GO] 2022―Apr―04 HIV protease inhibitors Nelfinavir and Lopinavir/Ritonavir markedly improve lung pathology in SARS-CoV-2-infected Syrian hamsters despite lack of an antiviral effect Caroline S. Foo, Rana Abdelnabi, Suzanne J.F. Kaptein, Xin Zhang, Sebastiaan ter Horst, Raf Mols, Leen Delang, Joana Rocha-Pereira, Lotte Coelmont, Pieter Leyssen, Kai Dallmeier, Valentijn Vergote, Elisabeth Heylen, Laura Vangeel, Arnab K. Chatterjee, Pieter P. Annaert, Patrick F. Augustijns, Steven De Jonghe, Dirk Jochmans, Mieke Gouwy, Seppe Cambier, Jennifer Vandooren, Paul Proost, Christine van Laer, Birgit Weynand, Johan Neyts
111 [GO] 2022―Mar―24 Isolation of human monoclonal antibodies with neutralizing activity to a broad spectrum of SARS-CoV-2 viruses including the Omicron variants Mikako Ueno, Naoko Iwata-Yoshikawa, Akihito Matsunaga, Tadashi Okamura, Sho Saito, Shinobu Ashida, Isao Yoshida, Mami Nagashima, Hiroyuki Asakura, Yuu I. Yaoita, Jun Suzuki, Kenji Sadamasu, Kazuhisa Yoshimura, Satoshi Kutsuna, Nozomi Shiwa-Sudo, Noriyo Nagata, Tadaki Suzuki, Akinori Suzuki, Miwa Okamoto, Moto Kimura, Norio Ohmagari, Ryu Miura, Yukihito Ishizaka
112 [GO] 2022―Mar―13 Neutralization or enhancement of SARS-CoV-2 infection by a monoclonal antibody targeting a specific epitope in the spike receptor-binding domain Guan-Chun Lai, Tai-Ling Chao, Shiau-Yu Lin, Han-Chieh Kao, Ya-Min Tsai, De-Chao Lu, Yi-Wei Chiang, Sui-Yuan Chang, Shih-Chung Chang
113 [GO] 2022―Mar―11 Novel antiviral activity of PAD inhibitors against human beta-coronaviruses HCoV-OC43 and SARS-CoV-2 Selina Pasquero, Francesca Gugliesi, Gloria Griffante, Valentina Dell’Oste, Matteo Biolatti, Camilla Albano, Greta Bajetto, Serena Delbue, Lucia Signorini, Maria Dolci, Santo Landolfo, Marco De Andrea
114 [GO] 2022―Mar―09 Label-free duplex SAMDI-MS screen reveals novel SARS-CoV-2 3CLpro inhibitors. M.D. Scholle, P. O'Kane, S. Dib, Z.A. Gurard-Levin
115 [GO] 2022―Mar―09 A highly sensitive cell-based luciferase assay for high-throughput automated screening of SARS-CoV-2 nsp5/3CLpro inhibitors K.Y. Chen, T. Krischuns, L.Ortega Varga, E. Harigua-Souiai, S. Paisant, A. Zettor, J. Chiaravalli, A. Delpal, D. Courtney, A. O'Brien, S.C. Baker, E. Decroly, C. Isel, F. Agou, Y. Jacob, A. Blondel, N. Naffakh
116 [GO] 2022―Mar―07 Establishment of a stable SARS-CoV-2 replicon system for application in high-throughput screening Tomohisa Tanaka, Akatsuki Saito, Tatsuya Suzuki, Yoichi Miyamoto, Kazuo Takayama, Toru Okamoto, Kohji Moriishi
117 [GO] 2022―Feb―28 ACE2-Fc fusion protein overcomes viral escape by potently neutralizing SARS-CoV-2 variants of concern Tsung-I Tsai, Jahan S. Khalili, Mark Gilchrist, Andrew B. Waight, Daniella Cohen, Shi Zhuo, Yong Zhang, Muran Ding, Hai Zhu, Amanda Nga-Sze Mak, Yi Zhu, Dennis R. Goulet
118 [GO] 2022―Jan―29 5-Iodotubercidin inhibits SARS-CoV-2 RNA synthesis Jianyuan Zhao, Qian Liu, Dongrong Yi, Quanjie Li, SaiSai Guo, Ling Ma, Yongxin Zhang, Dongxin Dong, Fei Guo, Zhenlong Liu, Tao Wei, Xiaoyu Li, Shan Cen
119 [GO] 2022―Jan―24 Remdesivir, Molnupiravir and Nirmatrelvir remain active against SARS-CoV-2 Omicron and other variants of concern Laura Vangeel, Winston Chiu, Steven De Jonghe, Piet Maes, Bram Slechten, Joren Raymenants, Emmanuel André, Pieter Leyssen, Johan Neyts, Dirk Jochmans
120 [GO] 2022―Jan―21 The omicron (B.1.1.529) SARS-CoV-2 variant of concern does not readily infect Syrian hamsters Rana Abdelnabi, Caroline S. Foo, Xin Zhang, Viktor Lemmens, Piet Maes, Bram Slechten, Joren Raymenants, Emmanuel André, Birgit Weynand, Kai Dallemier, Johan Neyts
121 [GO] 2022―Jan―13 Very low levels of remdesivir resistance in SARS-COV-2 genomes after 18 months of massive usage during the COVID19 pandemic: A GISAID exploratory analysis Daniele Focosi, Fabrizio Maggi, Scott McConnell, Arturo Casadevall
122 [GO] 2022―Jan―13 Subcutaneous remdesivir administration prevents interstitial pneumonia in rhesus macaques inoculated with SARS-CoV-2 Brandi N. Williamson, Lizzette Pérez-Pérez, Benjamin Schwarz, Friederike Feldmann, Myndi G. Holbrook, Manmeet Singh, Diane S. Lye, Darius Babusis, Raju Subramanian, Elaine Haddock, Atsushi Okumura, Patrick W. Hanley, Jamie Lovaglio, Catharine M. Bosio, Danielle P. Porter, Tomas Cihlar, Richard L. Mackman, Greg Saturday, Emmie de Wit
123 [GO] 2021―Dec―29 S-adenosylmethionine-dependent methyltransferase inhibitor DZNep blocks transcription and translation of SARS-CoV-2 genome with a low tendency to select for drug-resistant viral variants Ram Kumar, Nitin Khandelwal, Yogesh Chander, Himanshu Nagori, Assim Verma, Aditya Barua, Bhagraj Godara, Yash Pal, Baldev R. Gulati, Bhupendra N. Tripathi, Sanjay Barua, Naveen Kumar
124 [GO] 2021―Dec―18 COVID-19, Influenza and RSV: Surveillance-informed prevention and treatment - Meeting report from an isirv-WHO virtual conference Jennifer L. McKimm-Breschkin, Alan J. Hay, Bin Cao, Rebecca J. Cox, Jake Dunning, Ann C. Moen, Daniel Olsen, Andrés Pizzorno, Frederick G. Hayden
125 [GO] 2021―Nov―24 Hydroxychloroquine and azithromycin used alone or combined are not effective against SARS-CoV-2 ex vivo and in a hamster model Maxime Cochin, Franck Touret, Jean-Sélim Driouich, Gregory Moureau, Paul-Rémi Petit, Caroline Laprie, Caroline Solas, Xavier de Lamballerie, Antoine Nougairède
126 [GO] 2021―Nov―18 2-((1H-indol-3-yl)thio)-N-phenyl-acetamides: SARS-CoV-2 RNA-dependent RNA polymerase inhibitors Jianyuan Zhao, Guoning Zhang, Yongxin Zhang, Dongrong Yi, Quanjie Li, Ling Ma, SaiSai Guo, Xiaoyu Li, Fei Guo, Rongtuan Lin, Gia Luu, Zhenlong Liu, Yucheng Wang, Shan Cen
127 [GO] 2021―Nov―10 Picomolar inhibition of SARS-CoV-2 variants of concern by an engineered ACE2-IgG4-Fc fusion protein Hristo L. Svilenov, Julia Sacherl, Alwin Reiter, Lisa S. Wolff, Cho-Chin Cheng, Marcel Stern, Vincent Grass, Martin Feuerherd, Frank-Peter Wachs, Nicole Simonavicius, Susanne Pippig, Florian Wolschin, Oliver T. Keppler, Johannes Buchner, Carsten Brockmeyer, Ulrike Protzer
128 [GO] 2021―Nov―08 Development and characterization of SARS-CoV-2 variant-neutralizing monoclonal antibodies Hongyu Qiu, Xin-Yong Yuan, Teresa Cabral, Kathy Manguiat, Alyssia Robinson, Heidi Wood, Chris Grant, Peter McQueen, Garrett Westmacott, Daniel R. Beniac, Lisa Lin, Michael Carpenter, Darwyn Kobasa, Tom Gräfenhan
129 [GO] 2021―Oct―21 Inhibition of endocytosis of porcine reproductive and respiratory syndrome virus by rottlerin and its potential prophylactic administration in piglets Yeong-Lim Kang, Changin Oh, So-Hyun Ahn, Jong-Chul Choi, Hwi-Yeon Choi, Sang-Won Lee, In-Soo Choi, Chang-Seon Song, Joong-Bok Lee, Seung-Yong Park
130 [GO] 2021―Oct―08 SARS-CoV-2 monoclonal antibodies with therapeutic potential: Broad neutralizing activity and No evidence of antibody-dependent enhancement Ying-Ting Wang, Robert D. Allen, Kenneth Kim, Norazizah Shafee, Andrew J. Gonzalez, Michael N. Nguyen, Kristen M. Valentine, Xia Cao, Lucy Lu, Chin-I Pai, Sachi Johnson, Lisa Kerwin, Heyue Zhou, Yanliang Zhang, Sujan Shresta
131 [GO] 2021―Oct―07 A fluorescence-based, gain-of-signal, live cell system to evaluate SARS-CoV-2 main protease inhibition Rama Dey-Rao, George R. Smith, Uddhav Timilsina, Zackary Falls, Ram Samudrala, Spyridon Stavrou, Thomas Melendy
132 [GO] 2021―Aug―24 Identification of Niemann-Pick C1 protein as a potential novel SARS-CoV-2 intracellular target Isabel García-Dorival, Miguel Ángel Cuesta-Geijo, Lucía Barrado-Gil, Inmaculada Galindo, Urtzi Garaigorta, Jesús Urquiza, Ana del Puerto, Nuria E. Campillo, Ana Martínez, Pablo Gastaminza, Carmen Gil, Covadonga Alonso
133 [GO] 2021―Aug―09 Polyphenylene carboxymethylene (PPCM) microbicide repurposed as antiviral against SARS-CoV-2. Proof of concept in primary human undifferentiated epithelial cells Olivier Escaffre, Alexander N. Freiberg
134 [GO] 2021―Aug―08 A tetrameric ACE2 protein broadly neutralizes SARS-CoV-2 spike variants of concern with elevated potency Adam Leach, F. Tudor Ilca, Zulaikha Akbar, Mathieu Ferrari, Emma M. Bentley, Giada Mattiuzzo, Shimobi Onuoha, Ami Miller, Hanif Ali, Terence H. Rabbitts
135 [GO] 2021―Jul―23 Identification and evaluation of potential SARS-CoV-2 antiviral agents targeting mRNA cap guanine N7-Methyltransferase Renata Kasprzyk, Tomasz J. Spiewla, Miroslaw Smietanski, Sebastian Golojuch, Laura Vangeel, Steven De Jonghe, Dirk Jochmans, Johan Neyts, Joanna Kowalska, Jacek Jemielity
136 [GO] 2021―Jul―12 Preclinical evaluation of Imatinib does not support its use as an antiviral drug against SARS-CoV-2 Franck Touret, Jean-Sélim Driouich, Maxime Cochin, Paul Rémi Petit, Magali Gilles, Karine Barthélémy, Grégory Moureau, Francois-Xavier Mahon, Denis Malvy, Caroline Solas, Xavier de Lamballerie, Antoine Nougairède
137 [GO] 2021―Jul―08 A mouse model of lethal respiratory dysfunction for SARS-CoV-2 infection Esther S. Gan, Ayesa Syenina, Martin Linster, Benson Ng, Summer L. Zhang, Satoru Watanabe, Ravisankar Rajarethinam, Hwee Cheng Tan, Gavin JD. Smith, Eng Eong Ooi
138 [GO] 2021―Jun―26 A robust SARS-CoV-2 replication model in primary human epithelial cells at the air liquid interface to assess antiviral agents Thuc Nguyen Dan Do, Kim Donckers, Laura Vangeel, Arnab K. Chatterjee, Philippe A. Gallay, Michael D. Bobardt, John P. Bilello, Tomas Cihlar, Steven De Jonghe, Johan Neyts, Dirk Jochmans
139 [GO] 2021―Jun―19 Selinexor, a novel selective inhibitor of nuclear export, reduces SARS-CoV-2 infection and protects the respiratory system in vivo Trinayan Kashyap, Jackelyn Murray, Christopher J. Walker, Hua Chang, Sharon Tamir, Bing Hou, Sharon Shacham, Michael G. Kauffman, Ralph A. Tripp, Yosef Landesman
140 [GO] 2021―May―16 Virucidal and antiviral activity of astodrimer sodium against SARS-CoV-2 in vitro Jeremy R.A. Paull, Graham P. Heery, Michael D. Bobardt, Alex Castellarnau, Carolyn A. Luscombe, Jacinth K. Fairley, Philippe A. Gallay
141 [GO] 2021―Apr―21 A cell-based assay to discover inhibitors of SARS-CoV-2 RNA dependent RNA polymerase Jianyuan Zhao, SaiSai Guo, Dongrong Yi, Quanjie Li, Ling Ma, Yongxin Zhang, Jing Wang, Xiaoyu Li, Fei Guo, Rongtuan Lin, Chen Liang, Zhenlong Liu, Shan Cen
142 [GO] 2021―Apr―17 Discovery of Chebulagic Acid and Punicalagin as Novel Allosteric Inhibitors of SARS-CoV-2 3CLpro Ruikun Du, Laura Cooper, Zinuo Chen, Hyun Lee, Lijun Rong, Qinghua Cui
143 [GO] 2021―Mar―27 Proteomic Analysis Identifies the RNA Helicase DDX3X as a Host Target Against SARS-CoV-2 Infection Fabiola Ciccosanti, Martina Di Rienzo, Alessandra Romagnoli, Francesca Colavita, Giulia Refolo, Concetta Castilletti, Chiara Agrati, Annalaura Brai, Fabrizio Manetti, Lorenzo Botta, Maria Rosaria Capobianchi, Giuseppe Ippolito, Mauro Piacentini, Gian Maria Fimia
144 [GO] 2021―Mar―11 Emetine suppresses SARS-CoV-2 replication by inhibiting interaction of viral mRNA with eIF4E Ram Kumar, Mohammad Afsar, Nitin Khandelwal, Yogesh Chander, Thachamvally Riyesh, Ramesh Kumar Dedar, Baldev R. Gulati, Yash Pal, Sanjay Barua, Bhupendra N. Tripathi, Tanweer Hussain, Naveen Kumar
145 [GO] 2021―Mar―11 Combined in silico and in vitro approaches identified the antipsychotic drug lurasidone and the antiviral drug elbasvir as SARS-CoV2 and HCoV-OC43 inhibitors Mario Milani, Manuela Donalisio, Rafaela Milan Bonotto, Edoardo Schneider, Irene Arduino, Francesco Boni, David Lembo, Alessandro Marcello, Eloise Mastrangelo
146 [GO] 2021―Feb―06 Genetic Conservation of SARS-CoV-2 RNA Replication Complex in Globally Circulating Isolates and Recently Emerged Variants from Humans and Minks Suggests Minimal Pre-Existing Resistance to Remdesivir Ross Martin, Jiani Li, Aiyippa Parvangada, Jason Perry, Tomas Cihlar, Hongmei Mo, Danielle Porter, Evguenia Svarovskaia
147 [GO] 2021―Jan―27 Dual Inhibition of SARS-CoV-2 and Human Rhinovirus with Protease Inhibitors in Clinical Development Cheng Liu, Sandro Boland, Michael D. Scholle, Dorothee Bardiot, Arnaud Marchand, Patrick Chaltin, Lawrence M. Blatt, Leonid Beigelman, Julian A. Symons, Pierre Raboisson, Zachary A. Gurard-Levin, Koen Vandyck, Jerome Deval
148 [GO] 2021―Jan―13 Inhibition of coronavirus infection by a synthetic STING agonist in primary human airway system Qingyuan Zhu, Yaling Zhang, Li Wang, Xiangyu Yao, Daitze Wu, Junjun Cheng, Xiaoyu Pan, Haixia Liu, Zhipeng Yan, Lu Gao
149 [GO] 2021―Jan―08 The rocaglate CR-31-B (-) inhibits SARS-CoV-2 replication at non-cytotoxic, low nanomolar concentrations in vitro and ex vivo Christin Müller, Wiebke Obermann, Nadja Karl, Hans-Guido Wendel, Gaspar Taroncher-Oldenburg, Stephan Pleschka, Roland K. Hartmann, Arnold Grünweller, John Ziebuhr
150 [GO] 2020―Dec―10 Antiviral activity against Middle East Respiratory Syndrome Coronavirus by Montelukast, an anti-asthma drug Hanjie Jonathan Gan, Amaravadhi Harikishore, Jihye Lee, Sangeun Jeon, Sreekanth Rajan, Ming Wei Chen, Jun Long Neo, Seungtaek Kim, Ho Sup Yoon
151 [GO] 2020―Nov―25 Ionophore antibiotic X-206 is a potent inhibitor of SARS-CoV-2 infection in vitro Esben B. Svenningsen, Jacob Thyrsted, Julia Blay-Cadanet, Han Liu, Shaoquan Lin, Jaime Moyano Villameriel, David Olagnier, Manja Idorn, Søren R. Paludan, Christian K. Holm, Thomas B. Poulsen
152 [GO] 2020―Nov―17 A bacterial artificial chromosome (BAC)-vectored noninfectious replicon of SARS-CoV-2 Yang Zhang, Wuhui Song, Shuiye Chen, Zhenghong Yuan, Zhigang Yi
153 [GO] 2020―Oct―19 Antiviral activity and safety of remdesivir against SARS-CoV-2 infection in human pluripotent stem cell-derived cardiomyocytes Seong Woo Choi, Jin Soo Shin, Soon-Jung Park, Eunhye Jung, Yun-Gwi Park, Jiho Lee, Sung Joon Kim, Hun-Jun Park, Jung-Hoon Lee, Sung-Min Park, Sung-Hwan Moon, Kiwon Ban, Yun Young Go
154 [GO] 2020―Sep―19 Cryptotanshinone Protects Porcine Alveolar Macrophages from Infection with Porcine Reproductive and Respiratory Syndrome Virus Chang Huang, Jiaqi Zhu, Ling Wang, Alexander Chu, Yexuan Yin, Kaneha Vali, Antonio Garmendia, Young Tang
155 [GO] 2020―Sep―07 Structural-based virtual screening and in vitro assays for small molecules inhibiting the feline coronavirus 3CL protease as a surrogate platform for coronaviruses Sirin Theerawatanasirikul, Chih Jung Kuo, Nanthawan Phecharat, Jullada Chootip, Chalermpol Lekcharoensuk, Porntippa Lekcharoensuk
156 [GO] 2020―Sep―06 Evaluation of SARS-CoV-2 3C-like protease inhibitors using self-assembled monolayer desorption ionization mass spectrometry Zachary A. Gurard-Levin, Cheng Liu, Andreas Jekle, Ruchika Jaisinghani, Suping Ren, Koen Vandyck, Dirk Jochmans, Pieter Leyssen, Johan Neyts, Lawrence M. Blatt, Leonid Beigelman, Julian A. Symons, Pierre Raboisson, Michael D. Scholle, Jerome Deval
157 [GO] 2020―Jul―30 The chemokine receptor antagonist cenicriviroc inhibits the replication of SARS-CoV-2 in vitro Mika Okamoto, Masaaki Toyama, Masanori Baba
158 [GO] 2020―Jul―29 An enzyme-based immunodetection assay to quantify SARS-CoV-2 infection Carina Conzelmann, Andrea Gilg, Rüdiger Groß, Desiree Schütz, Nico Preising, Ludger Ständker, Bernd Jahrsdörfer, Hubert Schrezenmeier, Konstantin M.J. Sparrer, Thomas Stamminger, Steffen Stenger, Jan Münch, Janis A. Müller
159 [GO] 2020―Jul―15 In vitro evaluation of antiviral activity of single and combined repurposable drugs against SARS-CoV-2 Andrés Pizzorno, Blandine Padey, Julia Dubois, Thomas Julien, Aurélien Traversier, Victoria Dulière, Pauline Brun, Bruno Lina, Manuel Rosa-Calatrava, Olivier Terrier
160 [GO] 2020―Jul―15 Lower prevalence of antibodies neutralizing SARS-CoV-2 in group O French blood donors Pierre Gallian, Boris Pastorino, Pascal Morel, Jacques Chiaroni, Laetitia Ninove, Xavier de Lamballerie
161 [GO] 2020―Jul―10 Concerns about pharmacokinetic (PK) and pharmacokinetic-pharmacodynamic (PK-PD) studies in the new therapeutic area of COVID-19 infection Nicolas Venisse, Gilles Peytavin, Stephane Bouchet, Marie-Claude Gagnieu, Rodolphe Garraffo, Romain Guilhaumou, Caroline Solas
162 [GO] 2020―Jul―10 Characterization of heparin and severe acute respiratory syndrome-related coronavirus 2 (SARS-CoV-2) spike glycoprotein binding interactions So Young Kim, Weihua Jin, Amika Sood, David W. Montgomery, Oliver C. Grant, Mark M. Fuster, Li Fu, Jonathan S. Dordick, Robert J. Woods, Fuming Zhang, Robert J. Linhardt
163 [GO] 2020―Jul―10 Immunoglobulin fragment F(ab’)2 against RBD potently neutralizes SARS-CoV-2 in vitro Xiaoyan Pan, Pengfei Zhou, Tiejiong Fan, Yan Wu, Jing Zhang, Xiaoyue Shi, Weijuan Shang, Lijuan Fang, Xiaming Jiang, Jian Shi, Yuan Sun, Shaojuan Zhao, Rui Gong, Ze Chen, Gengfu Xiao
164 [GO] 2020―Jun―19 The influence of interferon-lambda on restricting Middle East Respiratory Syndrome Coronavirus replication in the respiratory epithelium Yung Jin Jeon, Chan Hee Gil, Ara Jo, Jina Won, Sujin Kim, Hyun Jik Kim
165 [GO] 2020―Jun―18 A Library of Nucleotide Analogues Terminate RNA Synthesis Catalyzed by Polymerases of Coronaviruses that Cause SARS and COVID-19 Steffen Jockusch, Chuanjuan Tao, Xiaoxu Li, Thomas K. Anderson, Minchen Chien, Shiv Kumar, James J. Russo, Robert N. Kirchdoerfer, Jingyue Ju
166 [GO] 2020―May―13 Identification of SARS-CoV RBD-targeting monoclonal antibodies with cross-reactive or neutralizing activity against SARS-CoV-2 Wanbo Tai, Xiujuan Zhang, Yuxian He, Shibo Jiang, Lanying Du
167 [GO] 2020―Apr―29 Antiviral Activities of Type I Interferons to SARS-CoV-2 Infection Emily Mantlo, Natalya Bukreyeva, Junki Maruyama, Slobodan Paessler, Cheng Huang
168 [GO] 2020―Apr―21 Ivermectin and COVID-19: a report in Antiviral Research, widespread interest, an FDA warning, two letters to the editor and the authors' responses Mike Bray, Craig Rayner, François Noël, David Jans, Kylie Wagstaff
169 [GO] 2020―Apr―10 Remdesivir and SARS-CoV-2: Structural requirements at both nsp12 RdRp and nsp14 Exonuclease active-sites Ashleigh Shannon, Nhung Thi-Tuyet Le, Barbara Selisko, Cecilia Eydoux, Karine Alvarez, Jean-Claude Guillemot, Etienne Decroly, Olve Peersen, Francois Ferron, Bruno Canard
170 [GO] 2020―Apr―07 Type 1 interferons as a potential treatment against COVID-19 Erwan Sallard, François-Xavier Lescure, Yazdan Yazdanpanah, France Mentre, Nathan Peiffer-Smadja
171 [GO] 2020―Apr―06 Coronavirus membrane fusion mechanism offers as a potential target for antiviral development Tiffany Tang, Miya Bidon, Javier A. Jaimes, Gary R. Whittaker, Susan Daniel
172 [GO] 2020―Apr―03 The FDA-approved Drug Ivermectin inhibits the replication of SARS-CoV-2 in vitro Leon Caly, Julian D. Druce, Mike G. Catton, David A. Jans, Kylie M. Wagstaff
173 [GO] 2020―Apr―03 Remdesivir, lopinavir, emetine, and homoharringtonine inhibit SARS-CoV-2 replication in vitro Ka-Tim Choy, Alvina Yin-Lam Wong, Prathanporn Kaewpreedee, Sin-Fun Sia, Dongdong Chen, Kenrie Pui Yan Hui, Daniel Ka Wing Chu, Michael Chi Wai Chan, Peter Pak-Hang Cheung, Xuhui Huang, Malik Peiris, Hui-Ling Yen
174 [GO] 2020―Mar―06 Of chloroquine and COVID-19 Franck Touret, Xavier de Lamballerie
175 [GO] 2020―Mar―01 A potential role for integrins in host cell entry by SARS-CoV-2 Christian JA Sigrist, Alan Bridge, Philippe Le Mercier
176 [GO] 2020―Feb―27 Efficacy of anti-influenza immunoglobulin (FLU-IGIV) in ferrets and mice infected with 2009 pandemic influenza virus Hongyu Qiu, Hanne Andersen, E. Bart Tarbet, F. Salih Muhammad, Trevor Carnelley, Russell Pronyk, Douglas Barker, Shantha Kodihalli
177 [GO] 2020―Feb―10 The spike glycoprotein of the new coronavirus 2019-nCoV contains a furin-like cleavage site absent in CoV of the same clade B. Coutard, C. Valle, X. de Lamballerie, B. Canard, N.G. Seidah, E. Decroly
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177 Results       Page 1



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